PepSight
MELANIN/SKIN

Melanotan-1 (Afamelanotide)

Melanotan-1 (Afamelanotide) is a melanin/skin peptide used in evidence-based, physician-supervised protocols. Use for photoprotection, tanning (aesthetic), and erythropoietic protoporphyria (FDA-approved in EU).

What is Melanotan-1 (Afamelanotide)?

Synthetic alpha-MSH analogue. Activates MC1R on melanocytes, driving melanin synthesis and increasing UV-induced melanogenesis. Safer profile than MT-II — does not activate MC3R/MC4R (no libido/erection effects). Loading phase: daily or EOD 2-4 weeks; maintenance: weekly.

Uses & clinical decision logic

Use for photoprotection, tanning (aesthetic), and erythropoietic protoporphyria (FDA-approved in EU).

Melanotan-1 (Afamelanotide) dosage & administration

Vial sizeBAC waterDosing rangeUnits / doseFrequencyRoute
10mg2mL250-500mcg5-10 unitsDaily or EOD (loading), Weekly (maintenance)SubQ

Safety & contraindications

Nausea common at initiation — start low (250mcg). Monitor skin lesions — do not use with atypical moles without dermatology clearance.

Stacking & combinations

Compatible with skin peptides (GHK-Cu, SNAP-8).

Related peptides

Frequently asked questions

What is Melanotan-1 (Afamelanotide) used for?

Use for photoprotection, tanning (aesthetic), and erythropoietic protoporphyria (FDA-approved in EU).

What is the typical Melanotan-1 (Afamelanotide) dosage?

Common dosing ranges from 250-500mcg (Daily or EOD (loading), Weekly (maintenance), SubQ). Exact dosing is individualized and set by a licensed physician.

How is Melanotan-1 (Afamelanotide) administered?

Melanotan-1 (Afamelanotide) is typically administered via SubQ.

What are the contraindications for Melanotan-1 (Afamelanotide)?

Nausea common at initiation — start low (250mcg). Monitor skin lesions — do not use with atypical moles without dermatology clearance.

Considering Melanotan-1 (Afamelanotide)?

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This page is for educational purposes only and is not medical advice. Peptide therapies described here are provided under physician supervision through 503A compounding pharmacies. Many peptides are not FDA-approved for the uses described. Do not start, stop, or change any protocol without consulting a licensed physician.